Whole Pharmacology Classification: Adrenergic Antagonists Alpha Adrenergic Antagonists Alpha 1 Antagonists
Whole Pharmacology Classification: Adrenergic Antagonists Alpha Adrenergic Antagonists Alpha 1 Antagonists
Adrenergic Antagonists
Alpha Adrenergic Antagonists
Alpha 1 antagonists
Prazosin
Doxazosin
Terazosin
Tamsulosin
Alfuzosin
Indoramin
Urapidil
Alpha 2 Antagonists:
Yohimbine
Tolazoline
Alpha 1 And Alpha 2 Antagonists:
Phenoxybenzamine
Phentolamine
Beta Adrenergic Antagonists
Beta 1 And Beta 2 Antagonists
Propranolol
Pindolol
Penbutolol
Nadolol
Carteolol
Timolol
Sotalol
Beta 1 Antagonists
Acebutolol
Atenolol
Alprenolol
Betaxolol
Celiprolol
Metoprolol
Esmolol
Nebivolol
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Adrenergic Agonists
Direct action
Non-selective: drugs act on one or more receptors; these are
Adrenaline (almost all adrenergic receptors).
Noradrenaline (acts on α1, α2, β1).
Isoprenaline (acts on β1, β2, β3).
Dopamine (acts on α1, α2, β1, D1, D2).
Selective: drugs which act on a single receptor only; these are further
classified into
α selective & β selective.
α1 selective: Phenylephrine, Methoxamine, Midodrine, Oxymetazoline.
α2 selective: α-Methyl dopa, clonidine, brimonidine.
β1 selective: Dobutamine.
β2 selective: Salbutamol/Albuterol, Terbutaline, Salmeterol, Formoterol,
Pirbuterol.
Indirect action
Amphetamines
Cocaine
Methylenedioxymethamphetamine (MDMA)
Tyramine
Nicotine
Caffeine
Methylphenidate
Mixed action
Ephedrine
Pseudoephedrine
Cholinergic Agonists
Direct and indirect acting Agonists
Direct Acting Agonist Drugs:
Choline Esters
Acetylcholine
Methacholine
Carbachol
Bethanechol
Cholinomimetic alkaloids
Muscarine
Nicotine
Pilocarpine
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Lobeline
Indirect Acting Drugs:
Reversibly Acting:
Neostigmine
Physostigmine
Demecarium
Pyridostigmine
Ambenonium
Irreversible Acting:
Echothiophate
Parathione
Malathione
Tetra ethyl Pyrophosphate
Pharmacology Classification of Cholinergic Antagonists
Antimuscarinic agents
Atropine
Benztropine
Biperiden
Chlorpheniramine
Dicyclomine
Dimenhydrinate
Diphenhydramine
Doxepin
Doxylamine
Glycopyrrolate
Ipratropium
Orphenadrine
Oxitropium
Oxybutynin
Propantheline bromide
Tolterodine
Tiotropium
Trihexyphenidyl
Scopolamine
Solifenacin
Tropicamide
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Antinicotinic agents
Bupropion
Dextromethorphan
Doxacurium
Hexamethonium
Mecamylamine
Tubocurarine
Pharmacology Classification of Anti Anginal Drugs
Organic Nitrates
Nitriglycerin
Isosorbide Dinitrate
Isosorbide Mononitrate
Amyl nitrite
Calcium Channel Blockers
Dihydropyridine
Nifedipine
Nicardipine
Amlodipine
Nisoldipine
Nitrendipine
Nimodipine
Miscellaneous Drugs
Verapamil
Diltiazem
Bepridil
Beta Blockers
ß 1 + ß 2 Antagonists
Propranolol
Penbutolol
Sotalol
Pindolol
Timolol
ß 1 Selective Antagonist
Metoprolol
Atenolol
Esmolol
Acebutolo
Betaxolol
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Drugs used in Congestive cardiac failure
Drugs used to decrease preload:
Diuretics
Organic nitrate
Drugs which decrease after load
Hydralazine
Minoxidil
Drugs which decrease both preload and afterload:
Captopril
Enalapril
Lisinopril
Fosinopril
Quinapril
Positive ionotropic drugs:
Cardiac glycosides:
Digoxin
Digitoxin
Ouabin
Lanatoside.
Phosphodiestrase inhibitors:
Inamrinonone (Amrinone)
Milrinone
Sympathomimetics:
Dopamine
Dobutamine
Depoxamine
Xamoterol
Pharmacology Classification of Antiplatelet Drugs
Antiplatelet List of drugs include:
Anagrelide
Aspirin
Clopidogrel
Prasugrel
Ticagrelor
Tirofiban
Vorapaxar
Dipyridamole
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Anticoagulant Drugs
Warfarin
Dabigatran
Edoxaban
Rivaroxaban
Apixaban
Diuretics
Thiazides diuretics
Chlorothiazide
Chlorthalidone
Indapamide
Hydrochlorothiazide
Methyclothiazide
Metolazone
Loop diuretics
Bumetanide
Furosemide
Ethacrynate
Torsemide
Potassium sparing diuretics
Amiloride hydrochloride
Spironolactone
Triamterene
Pharmacology Classification of Statins
Atorvastatin
Fluvastatin
Lovastatin
Pravastatin
Rosuvastatin
Simvastatin
Pitavastatin
Thrombolytic Drug
Anistreplase
Reteplase
Streptokinase, kabikinase
t-PA (class of drugs that includes Activase)
TNKase (tenecteplase)
Abbokinase, Kinlytic (rokinase)
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Pharmacology Classification of Sedative Hypnotic
Sedative Anxiolytic Drugs
Benzodiazepines
Alprazolam
Bromazepam
Chlordiazepoxide
Clonazepam
Clorazepate
Diazepam
Flurazepam
Lorazepam
Oxazepam
Temazepam
Triazolam
Barbiturates
Phenobarbital
Mephobarbital
Amobarbital sodium
Butabarbital sodium
Secobarbital sodium
Non Sedative
Buspirone
Gepirone
Ipsapirone
Tandospirone
Antidepressants
Tricyclic Antidepressant
Amitriptyline
Amoxapine
Desipramine
Doxepin
Imipramine
Nortriptyline
Protriptyline
Trimipramine
Selective serotonin reuptake inhibitors (SSRIs)
Citalopram
Escitalopram
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Paroxetine
Fluoxetine
Fluvoxamine
Sertraline
Serotonin–norepinephrine reuptake inhibitors (SNRIs)
Desvenlafaxine
Duloxetine
Levomilnacipran
Milnacipran
Venlafaxine
Serotonin modulators and stimulators (SMS)
Vilazodone
Vortioxetine
Norepinephrine reuptake inhibitors (NRIs)
Reboxetine
Teniloxazine
Viloxazine
Monoamine Oxidase Inhibitors
Isocarboxazid
Phenelzine
Selegiline
Tranylcypromine
Antipsychotic Drugs
Aripiprazole
Asenapine
Cariprazine
Clozapine
Lurasidone
Olanzapine
Quetiapine
Risperidone
Ziprasidone
Anti epileptic Drugs
Acetazolamide
Clonazepam
Ethosuximide
Lamotrigine
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Sodium valproate
Atonic seizures:
Phenobarbital
Phenytoin
Primidone
Sodium valproate
Catamenial seizures (menstrual-related):
Acetazolamide
Clobazam
Cluster seizures:
Clobazam
Episodic disorders:
Stiripentol
Focal (partial) seizures:
Acetazolamide
Carbamazepine
Clobazam
Clonazepam
Eslicarbazepine acetate
Gabapentin
Lacosamide
Lamotrigine
Levetiracetam
Oxcarbazepine
Perampanel
Phenobarbital
Phenytoin
Pregabalin
Primidone
Retigabine
Sodium valproate
Tiagabine
Topiramate
Vigabatrin
Zonisamide
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Focal (partial) seizures with secondary generalisation:
Gabapentin
Lacosamide
Levetiracetam
Perampanel
Phenobarbital
Phenytoin
Pregabalin
Primidone
Retigabine
Sodium valproate
Tiagabine
Topiramate
Vigabatrin
Zonisamide
Focal seizures with secondary generalised tonic clonic seizures:
Carbamazepine
Eslicarbazepine acetate
Lamotrigine
Oxcarbazepine
Infantile spasms:
Nitrazepam
Sodium valproate
Vigabatrin
Juvenile Myoclonic Epilepsy (seizures related to):
Levetiracetam
Lennox-Gastaut syndrome (seizures related to):
Lamotrigine
Rufinamide
Topiramate
Myoclonic seizures:
Clonazepam
Ethosuximide
Phenobarbital
Phenytoin
Primidone
Piracetam
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Sodium valproate
Tonic seizures:
Phenobarbital
Phenytoin
Primidone
Sodium valproate
Tonic clonic seizures:
Acetazolamide
Carbamazepine
Clobazam
Clonazepam
Eslicarbazepine acetate
Lamotrigine
Phenobarbital
Phenytoin
Primidone
Sodium valproate
Topiramate
West Syndrome with Tuberous Sclerosis:
Vigabatrin
Anesthetic Drugs
Local anesthetics
Procaine
Amethocaine
Lidocaine (also known as lignocaine)
Prilocaine
Bupivacaine
Levobupivacaine
Ropivacaine
Mepivacaine
Dibucaine
Cocaine
General anesthetics
Inhaled agents
Desflurane
Enflurane
Halothane
Isoflurane
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Methoxyflurane
Nitrous oxide
Sevoflurane
Xenon
Cocaine
Intravenous agents (non-opioid)
Barbiturates
Amobarbital (trade name: Amytal)
Methohexital (trade name: Brevital)
Thiamylal (trade name: Surital)
Thiopental
Benzodiazepines
Diazepam
Lorazepam
Midazolam
Etomidate
Ketamine
Propofol
Non Steroidal Anti-inflammatory Drugs
Aspirin
Celecoxib
Diclofenac
Diflunisal
Etodolac
Ibuprofen
Ketoprofen
Ketorolac
Nabumetone
Naproxen
Oxaprozin
Piroxicam
Disease Modifying Anti Rheumatic Drugs
Immunosuppressive Drugs
Methotrexate
Cyclophophamide
Azathioprine
Chlorambucil
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Cyclosporine
Mycophenolate mofetil
Leflunamide
Gold Compounds
Aurothiomalate
Aurothioglucose
Auranofin
Aminoquinolines
Chloroquine
Hydroxychloroquine alpha
Antigout Drugs
Drugs For the treatment of Acute Attack of Gout
Colchicine
NSAIDs
Drugs For the Prevention Of Gout
Uricosuric Drugs ( Probencid, Sulphinopyrazine
Inhibitors of Uric Acid synthesis (allopurinol, Febuxostat
Anti-migraine Drugs
Drugs For the Treatment OF Acute Attack
5-HT1 Agonists
Sumatriptan
Zolmitriptan
Naratriptan
Rizatriptan
Other Drugs
Ergotamine
Dihydroergotamine
NSAIDs
Paracetamol
Opioids
Prophylactic Drugs
Propranolol
Aspirin
Pizotifen
Cyproheptadine
Amitriptyline
Imipramine
Fluoxetine
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Sertraline
Methysergide
Flunarizine
Clonidine
Antimicrobial Drugs
Beta Lactam Antimicrobials
Penicillin
Cephalosporins
Monobactams
Carbaphenems
Penicillin Narrow Spectrum Penicillin
Penicillinase Sensitive Penicillin
Penicillin G (Benzyl Penicillin)
Penicillin V
Penicillinase Resistant Penicillin
Nafcillin
Oxacillin
Cloxacillin
Dicloxacillin
Flucloxacillin
Methicillin
Broad Spectrum Penicillin
Aminopenicillin
Ampicillin
Amoxicillin
Bacampicillin
Talampicillin
Antipseudomonal Penicillin
Carboxypenicillin
Carbencillin
Ticarcillin
Ureidopenicillins
Azlocillin
Mezlocillin
Piperacillin
Fluoroquinolones ;
First Generation e.g Nalidix acid
Second Generation e.g Ciprofloxacin,Norfloxacin and ofloxacin.
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Norfloxacin don’t absorb very well and they are not used most commonly
While ciprofloxacin is the most commonly used drug in this class.
Third Generation E.g Levofloxacin
Fourth Generation : Moxifloxacin
Cephalosporins
First-Generation Cephalosporins
Cefadroxil
Cefazedone
Cefazolin
Cephalexin
Cephalothin
Cephradine
Cephaloridine
Cephapirin
Second-Generation Cephalosporins
Cefaclor
Cefamandole
Cefprozil
Cefuroxime
Loracarbef
Third-Generation Cephalosporins
Cefcapene
Cefdinir
Cefditoren
Cefetamet
Cefixime
Cefmenoxime
Cefoperazone
Cefotaxime
Cefpiramide
Cefpodoxime
Cefsulodin
Ceftibuten
Ceftizoxime
Ceftriaxone
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Fourth-Generation Cephalosporins
Cefepime
Cefluprenam
Cefozopran
Cefpirome
Cefquinome
Sulfa Drugs
Co-Trimoxazole
Sulfadiazine
Sulfamethoxazole
Trimethoprim-Sulfamethoxazole
Trimethoprim
Sulfasalazine
Sulfisoxazole
Antitubercular Drugs
First Line Drugs
Isoniazid
Rifampicin
Pyrazinamide
Ethambutol
Streptomycin
Second Line Drugs
Para aminosalicylic Acid
Amikacin
Capreomycin
Ciprofloxacin
Clofazimine
Cycloserine
Ethionamide
Levofloxacin
Rifabutin
Rifapentine
Macrolide
Azithromycin
Clarithromycin
Erythromycin
Telithromycin
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Spiramycin
Laxative Drugs
Osmotic laxatives include the following:
Lactulose.
Glycerin.
Polyethylene glycol and electrolytes.
Glycerin rectal.
Polyethylene glycol electrolyte solution.
Polyethylene glycol powder.
Sodium sulfate/potassium sulfate/magnesium sulfate.
Polyethylene glycol/electrolytes/sodium ascorbate/ascorbic acid.
Milk of magnesia,
Magnesium citrate,
Sorbitol.
Antidiabetic Drugs
Biguanides like metformin.
Meglitinides like nateglinide and repaglinide
Sulfonylureas such as glimepiride, glipizide, glyburide, glyclazide and
tolazamide.
Thiazolidinediones (Tzd) such as pioglitazone, Actosgeneric and
rosiglitazone.
Alpha-glucosidase inhibitors like Acarbose.
Dopamine agonist such as Bromocriptine.
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