0% found this document useful (0 votes)
315 views

Whole Pharmacology Classification: Adrenergic Antagonists Alpha Adrenergic Antagonists Alpha 1 Antagonists

The document provides a classification of various types of pharmacology drugs organized into categories. It includes classifications for adrenergic drugs, cholinergic drugs, anti-anginal drugs, diuretics, statins, thrombolytic drugs, sedative-hypnotic drugs, antidepressants, antipsychotics, antiepileptics, anesthetics, NSAIDs, DMARDs, antigout drugs, antimigraine drugs, and antimicrobials. Each category lists the individual drug names under relevant subcategories.

Uploaded by

Florina Trutescu
Copyright
© © All Rights Reserved
We take content rights seriously. If you suspect this is your content, claim it here.
Available Formats
Download as DOCX, PDF, TXT or read online on Scribd
0% found this document useful (0 votes)
315 views

Whole Pharmacology Classification: Adrenergic Antagonists Alpha Adrenergic Antagonists Alpha 1 Antagonists

The document provides a classification of various types of pharmacology drugs organized into categories. It includes classifications for adrenergic drugs, cholinergic drugs, anti-anginal drugs, diuretics, statins, thrombolytic drugs, sedative-hypnotic drugs, antidepressants, antipsychotics, antiepileptics, anesthetics, NSAIDs, DMARDs, antigout drugs, antimigraine drugs, and antimicrobials. Each category lists the individual drug names under relevant subcategories.

Uploaded by

Florina Trutescu
Copyright
© © All Rights Reserved
We take content rights seriously. If you suspect this is your content, claim it here.
Available Formats
Download as DOCX, PDF, TXT or read online on Scribd
You are on page 1/ 17

Whole Pharmacology Classification

Adrenergic Antagonists
Alpha Adrenergic Antagonists
Alpha 1 antagonists
 Prazosin
 Doxazosin
 Terazosin
 Tamsulosin
 Alfuzosin
 Indoramin
 Urapidil
Alpha 2 Antagonists:
 Yohimbine
 Tolazoline
Alpha 1 And Alpha 2 Antagonists:
 Phenoxybenzamine
 Phentolamine
Beta Adrenergic Antagonists
Beta 1 And Beta 2 Antagonists
 Propranolol
 Pindolol
 Penbutolol
 Nadolol
 Carteolol
 Timolol
 Sotalol
Beta 1 Antagonists
 Acebutolol
 Atenolol
 Alprenolol
 Betaxolol
 Celiprolol
 Metoprolol
 Esmolol
 Nebivolol

1
Adrenergic Agonists
Direct action
Non-selective: drugs act on one or more receptors; these are
 Adrenaline (almost all adrenergic receptors).
 Noradrenaline (acts on α1, α2, β1).
 Isoprenaline (acts on β1, β2, β3).
 Dopamine (acts on α1, α2, β1, D1, D2).
Selective: drugs which act on a single receptor only; these are further
classified into
α selective & β selective.
 α1 selective: Phenylephrine, Methoxamine, Midodrine, Oxymetazoline.
 α2 selective: α-Methyl dopa, clonidine, brimonidine.
 β1 selective: Dobutamine.
 β2 selective: Salbutamol/Albuterol, Terbutaline, Salmeterol, Formoterol,
Pirbuterol.
Indirect action
 Amphetamines
 Cocaine
 Methylenedioxymethamphetamine (MDMA)
 Tyramine
 Nicotine
 Caffeine
 Methylphenidate
Mixed action
 Ephedrine
 Pseudoephedrine
Cholinergic Agonists
Direct and indirect acting Agonists
Direct Acting Agonist Drugs:
Choline Esters
 Acetylcholine
 Methacholine
 Carbachol
 Bethanechol
Cholinomimetic alkaloids
 Muscarine
 Nicotine
 Pilocarpine

2
 Lobeline
Indirect Acting Drugs:
Reversibly Acting:
 Neostigmine
 Physostigmine
 Demecarium
 Pyridostigmine
 Ambenonium
Irreversible Acting:
 Echothiophate
 Parathione
 Malathione
 Tetra ethyl Pyrophosphate
Pharmacology Classification of Cholinergic Antagonists
Antimuscarinic agents
 Atropine
 Benztropine
 Biperiden
 Chlorpheniramine
 Dicyclomine
 Dimenhydrinate
 Diphenhydramine
 Doxepin
 Doxylamine
 Glycopyrrolate
 Ipratropium
 Orphenadrine
 Oxitropium
 Oxybutynin
 Propantheline bromide
 Tolterodine
 Tiotropium
 Trihexyphenidyl
 Scopolamine
 Solifenacin
 Tropicamide

3
Antinicotinic agents
 Bupropion
 Dextromethorphan
 Doxacurium
 Hexamethonium
 Mecamylamine
 Tubocurarine
Pharmacology Classification of Anti Anginal Drugs
Organic Nitrates
 Nitriglycerin
 Isosorbide Dinitrate
 Isosorbide Mononitrate
 Amyl nitrite
Calcium Channel Blockers
Dihydropyridine
 Nifedipine
 Nicardipine
 Amlodipine
 Nisoldipine
 Nitrendipine
 Nimodipine
Miscellaneous Drugs
 Verapamil
 Diltiazem
 Bepridil
Beta Blockers
ß 1 + ß 2 Antagonists
 Propranolol
 Penbutolol
 Sotalol
 Pindolol
 Timolol
ß 1 Selective Antagonist
 Metoprolol
 Atenolol
 Esmolol
 Acebutolo
 Betaxolol
4
Drugs used in Congestive cardiac failure
Drugs used to decrease preload:
 Diuretics
 Organic nitrate
Drugs which decrease after load
 Hydralazine
 Minoxidil
Drugs which decrease both preload and afterload:
 Captopril
 Enalapril
 Lisinopril
 Fosinopril
 Quinapril
Positive ionotropic drugs:
Cardiac glycosides:
 Digoxin
 Digitoxin
 Ouabin
 Lanatoside.
Phosphodiestrase inhibitors:
 Inamrinonone (Amrinone)
 Milrinone
Sympathomimetics:
 Dopamine
 Dobutamine
 Depoxamine
 Xamoterol
Pharmacology Classification of Antiplatelet Drugs
Antiplatelet List of drugs include:
 Anagrelide
 Aspirin
 Clopidogrel
 Prasugrel
 Ticagrelor
 Tirofiban
 Vorapaxar
 Dipyridamole

5
Anticoagulant Drugs
 Warfarin
 Dabigatran
 Edoxaban
 Rivaroxaban
 Apixaban
Diuretics
Thiazides diuretics
 Chlorothiazide
 Chlorthalidone
 Indapamide
 Hydrochlorothiazide
 Methyclothiazide
 Metolazone
Loop diuretics
 Bumetanide
 Furosemide
 Ethacrynate
 Torsemide
Potassium sparing diuretics
 Amiloride hydrochloride
 Spironolactone
 Triamterene
Pharmacology Classification of Statins
 Atorvastatin
 Fluvastatin
 Lovastatin
 Pravastatin
 Rosuvastatin
 Simvastatin
 Pitavastatin
Thrombolytic Drug
 Anistreplase
 Reteplase
 Streptokinase, kabikinase
 t-PA (class of drugs that includes Activase)
 TNKase (tenecteplase)
 Abbokinase, Kinlytic (rokinase)
6
Pharmacology Classification of Sedative Hypnotic
Sedative Anxiolytic Drugs
 Benzodiazepines
 Alprazolam
 Bromazepam
 Chlordiazepoxide
 Clonazepam
 Clorazepate
 Diazepam
 Flurazepam
 Lorazepam
 Oxazepam
 Temazepam
 Triazolam
Barbiturates
 Phenobarbital
 Mephobarbital
 Amobarbital sodium
 Butabarbital sodium
 Secobarbital sodium
Non Sedative
 Buspirone
 Gepirone
 Ipsapirone
 Tandospirone
Antidepressants
Tricyclic Antidepressant
 Amitriptyline
 Amoxapine
 Desipramine
 Doxepin
 Imipramine
 Nortriptyline
 Protriptyline
 Trimipramine
Selective serotonin reuptake inhibitors (SSRIs)
 Citalopram
 Escitalopram
7
 Paroxetine
 Fluoxetine
 Fluvoxamine
 Sertraline
Serotonin–norepinephrine reuptake inhibitors (SNRIs)
 Desvenlafaxine
 Duloxetine
 Levomilnacipran
 Milnacipran
 Venlafaxine
Serotonin modulators and stimulators (SMS)
 Vilazodone
 Vortioxetine
Norepinephrine reuptake inhibitors (NRIs)
 Reboxetine
 Teniloxazine
 Viloxazine
Monoamine Oxidase Inhibitors
 Isocarboxazid
 Phenelzine
 Selegiline
 Tranylcypromine
Antipsychotic Drugs
 Aripiprazole
 Asenapine
 Cariprazine
 Clozapine
 Lurasidone
 Olanzapine
 Quetiapine
 Risperidone
 Ziprasidone
Anti epileptic Drugs
 Acetazolamide
 Clonazepam
 Ethosuximide
 Lamotrigine

8
 Sodium valproate
Atonic seizures:
 Phenobarbital
 Phenytoin
 Primidone
 Sodium valproate
Catamenial seizures (menstrual-related):
 Acetazolamide
 Clobazam
 Cluster seizures:
 Clobazam
Episodic disorders:
 Stiripentol
Focal (partial) seizures:
 Acetazolamide
 Carbamazepine
 Clobazam
 Clonazepam
 Eslicarbazepine acetate
 Gabapentin
 Lacosamide
 Lamotrigine
 Levetiracetam
 Oxcarbazepine
 Perampanel
 Phenobarbital
 Phenytoin
 Pregabalin
 Primidone
 Retigabine
 Sodium valproate
 Tiagabine
 Topiramate
 Vigabatrin
 Zonisamide

9
Focal (partial) seizures with secondary generalisation:
 Gabapentin
 Lacosamide
 Levetiracetam
 Perampanel
 Phenobarbital
 Phenytoin
 Pregabalin
 Primidone
 Retigabine
 Sodium valproate
 Tiagabine
 Topiramate
 Vigabatrin
 Zonisamide
Focal seizures with secondary generalised tonic clonic seizures:
 Carbamazepine
 Eslicarbazepine acetate
 Lamotrigine
 Oxcarbazepine
Infantile spasms:
 Nitrazepam
 Sodium valproate
 Vigabatrin
Juvenile Myoclonic Epilepsy (seizures related to):
 Levetiracetam
Lennox-Gastaut syndrome (seizures related to):
 Lamotrigine
 Rufinamide
 Topiramate
Myoclonic seizures:
 Clonazepam
 Ethosuximide
 Phenobarbital
 Phenytoin
 Primidone
 Piracetam

10
 Sodium valproate
Tonic seizures:
 Phenobarbital
 Phenytoin
 Primidone
 Sodium valproate
Tonic clonic seizures:
 Acetazolamide
 Carbamazepine
 Clobazam
 Clonazepam
 Eslicarbazepine acetate
 Lamotrigine
 Phenobarbital
 Phenytoin
 Primidone
 Sodium valproate
 Topiramate
West Syndrome with Tuberous Sclerosis:
 Vigabatrin
Anesthetic Drugs
Local anesthetics
 Procaine
 Amethocaine
 Lidocaine (also known as lignocaine)
 Prilocaine
 Bupivacaine
 Levobupivacaine
 Ropivacaine
 Mepivacaine
 Dibucaine
 Cocaine
General anesthetics
Inhaled agents
 Desflurane
 Enflurane
 Halothane
 Isoflurane
11
 Methoxyflurane
 Nitrous oxide
 Sevoflurane
 Xenon
 Cocaine
Intravenous agents (non-opioid)
Barbiturates
 Amobarbital (trade name: Amytal)
 Methohexital (trade name: Brevital)
 Thiamylal (trade name: Surital)
 Thiopental
Benzodiazepines
 Diazepam
 Lorazepam
 Midazolam
 Etomidate
 Ketamine
 Propofol
Non Steroidal Anti-inflammatory Drugs
 Aspirin
 Celecoxib
 Diclofenac
 Diflunisal
 Etodolac
 Ibuprofen
 Ketoprofen
 Ketorolac
 Nabumetone
 Naproxen
 Oxaprozin
 Piroxicam
Disease Modifying Anti Rheumatic Drugs
Immunosuppressive Drugs
 Methotrexate
 Cyclophophamide
 Azathioprine
 Chlorambucil

12
 Cyclosporine
 Mycophenolate mofetil
 Leflunamide
Gold Compounds
 Aurothiomalate
 Aurothioglucose
 Auranofin
Aminoquinolines
 Chloroquine
 Hydroxychloroquine alpha
Antigout Drugs
Drugs For the treatment of Acute Attack of Gout
 Colchicine
 NSAIDs
Drugs For the Prevention Of Gout
 Uricosuric Drugs ( Probencid, Sulphinopyrazine
 Inhibitors of Uric Acid synthesis (allopurinol, Febuxostat
Anti-migraine Drugs
Drugs For the Treatment OF Acute Attack
5-HT1 Agonists
 Sumatriptan
 Zolmitriptan
 Naratriptan
 Rizatriptan
Other Drugs
 Ergotamine
 Dihydroergotamine
 NSAIDs
 Paracetamol
 Opioids
Prophylactic Drugs
 Propranolol
 Aspirin
 Pizotifen
 Cyproheptadine
 Amitriptyline
 Imipramine
 Fluoxetine
13
 Sertraline
 Methysergide
 Flunarizine
 Clonidine
Antimicrobial Drugs
Beta Lactam Antimicrobials
 Penicillin
 Cephalosporins
 Monobactams
 Carbaphenems
Penicillin Narrow Spectrum Penicillin
Penicillinase Sensitive Penicillin
 Penicillin G (Benzyl Penicillin)
 Penicillin V
Penicillinase Resistant Penicillin
 Nafcillin
 Oxacillin
 Cloxacillin
 Dicloxacillin
 Flucloxacillin
 Methicillin
Broad Spectrum Penicillin
Aminopenicillin
 Ampicillin
 Amoxicillin
 Bacampicillin
 Talampicillin
Antipseudomonal Penicillin
Carboxypenicillin
 Carbencillin
 Ticarcillin
Ureidopenicillins
 Azlocillin
 Mezlocillin
 Piperacillin
Fluoroquinolones ;
 First Generation e.g Nalidix acid
 Second Generation e.g Ciprofloxacin,Norfloxacin and ofloxacin.
14
Norfloxacin don’t absorb very well and they are not used most commonly
While ciprofloxacin is the most commonly used drug in this class.
 Third Generation E.g Levofloxacin
 Fourth Generation : Moxifloxacin
Cephalosporins
First-Generation Cephalosporins
 Cefadroxil
 Cefazedone
 Cefazolin
 Cephalexin
 Cephalothin
 Cephradine
 Cephaloridine
 Cephapirin
Second-Generation Cephalosporins
 Cefaclor
 Cefamandole
 Cefprozil
 Cefuroxime
 Loracarbef
Third-Generation Cephalosporins
 Cefcapene
 Cefdinir
 Cefditoren
 Cefetamet
 Cefixime
 Cefmenoxime
 Cefoperazone
 Cefotaxime
 Cefpiramide
 Cefpodoxime
 Cefsulodin
 Ceftibuten
 Ceftizoxime
 Ceftriaxone

15
Fourth-Generation Cephalosporins
 Cefepime
 Cefluprenam
 Cefozopran
 Cefpirome
 Cefquinome
Sulfa Drugs
 Co-Trimoxazole
 Sulfadiazine
 Sulfamethoxazole
 Trimethoprim-Sulfamethoxazole
 Trimethoprim
 Sulfasalazine
 Sulfisoxazole
Antitubercular Drugs
First Line Drugs
 Isoniazid
 Rifampicin
 Pyrazinamide
 Ethambutol
 Streptomycin
Second Line Drugs
 Para aminosalicylic Acid
 Amikacin
 Capreomycin
 Ciprofloxacin
 Clofazimine
 Cycloserine
 Ethionamide
 Levofloxacin
 Rifabutin
 Rifapentine
Macrolide
 Azithromycin
 Clarithromycin
 Erythromycin
 Telithromycin

16
 Spiramycin
Laxative Drugs
Osmotic laxatives include the following:
 Lactulose.
 Glycerin.
 Polyethylene glycol and electrolytes.
 Glycerin rectal.
 Polyethylene glycol electrolyte solution.
 Polyethylene glycol powder.
 Sodium sulfate/potassium sulfate/magnesium sulfate.
 Polyethylene glycol/electrolytes/sodium ascorbate/ascorbic acid.
 Milk of magnesia,
 Magnesium citrate,
 Sorbitol.
Antidiabetic Drugs
 Biguanides like metformin.
 Meglitinides like nateglinide and repaglinide
 Sulfonylureas such as glimepiride, glipizide, glyburide, glyclazide and
tolazamide.
 Thiazolidinediones (Tzd) such as pioglitazone, Actosgeneric and
rosiglitazone.
 Alpha-glucosidase inhibitors like Acarbose.
 Dopamine agonist such as Bromocriptine.

17

You might also like

pFad - Phonifier reborn

Pfad - The Proxy pFad of © 2024 Garber Painting. All rights reserved.

Note: This service is not intended for secure transactions such as banking, social media, email, or purchasing. Use at your own risk. We assume no liability whatsoever for broken pages.


Alternative Proxies:

Alternative Proxy

pFad Proxy

pFad v3 Proxy

pFad v4 Proxy