The c-MYC oncoprotein is a substrate of the acetyltransferases hGCN5/PCAF and TIP60

Mol Cell Biol. 2004 Dec;24(24):10826-34. doi: 10.1128/MCB.24.24.10826-10834.2004.

Abstract

The c-MYC oncoprotein functions as a sequence-specific transcription factor. The ability of c-MYC to activate transcription relies in part on the recruitment of cofactor complexes containing the histone acetyltransferases mammalian GCN5 (mGCN5)/PCAF and TIP60. In addition to acetylating histones, these enzymes have been shown to acetylate other proteins involved in transcription, including sequence-specific transcription factors. This study was initiated in order to determine whether c-MYC is a direct substrate of mGCN5 and TIP60. We report here that mGCN5/PCAF and TIP60 acetylate c-MYC in vivo. By using nanoelectrospray tandem mass spectrometry to examine c-MYC purified from human cells, the major mGCN5-induced acetylation sites have been mapped. Acetylation of c-MYC by either mGCN5/PCAF or TIP60 results in a dramatic increase in protein stability. The data reported here suggest a conserved mechanism by which acetyltransferases regulate c-MYC function by altering its rate of degradation.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Acetylation
  • Acetyltransferases / metabolism*
  • Amino Acid Sequence
  • Blotting, Western
  • Cell Cycle Proteins / metabolism*
  • Cell Line, Tumor
  • Half-Life
  • Histone Acetyltransferases
  • Humans
  • Lung Neoplasms / pathology
  • Lysine Acetyltransferase 5
  • Precipitin Tests
  • Protein Structure, Tertiary
  • Proto-Oncogene Proteins c-myc / chemistry
  • Proto-Oncogene Proteins c-myc / genetics
  • Proto-Oncogene Proteins c-myc / metabolism*
  • Sequence Deletion
  • Substrate Specificity
  • Trans-Activators / metabolism*
  • Transcription Factors / genetics
  • Transcription Factors / metabolism*
  • p300-CBP Transcription Factors

Substances

  • Cell Cycle Proteins
  • Proto-Oncogene Proteins c-myc
  • Trans-Activators
  • Transcription Factors
  • Acetyltransferases
  • Histone Acetyltransferases
  • KAT2A protein, human
  • KAT5 protein, human
  • Lysine Acetyltransferase 5
  • p300-CBP Transcription Factors
  • p300-CBP-associated factor
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